SCHEMBL28520375

SCHEMBL28520375

O=C(NN=Cc1ccc(O)cc1O)c1cc([N+](=O)[O-])cc([N+](=O)[O-])c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DUSP3 P51452 1/20 0.62
PTPN5 P54829 1/20 0.62
PTPN11 Q06124 1/20 0.62
MEN1 O00255 5/20 0.62
KMT2A Q03164 5/20 0.62
NPC1 O15118 1/20 0.62
RAB9A P51151 1/20 0.62
PHGDH O43175 1/20 0.61
KDM4E B2RXH2 4/20 0.60
MAPT P10636 4/20 0.60
LMNA P02545 3/20 0.60
TDP1 Q9NUW8 3/20 0.60
ALDH1A1 P00352 3/20 0.60
SIRT1 Q96EB6 1/20 0.59
L3MBTL1 Q9Y468 2/20 0.58
ALPL P05186 1/20 0.58
POLB P06746 1/20 0.58
ALPI P09923 1/20 0.58
ALPG P10696 1/20 0.58
EIF4H Q15056 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28508004 0.90 MEN1 (0.73) DUSP3PTPN5PTPN11MEN1KMT2A
SCHEMBL28510646 0.89 DUSP3 (0.79) DUSP3PTPN5PTPN11MEN1KMT2A
SCHEMBL17988189 0.86 DUSP3 (0.82) DUSP3PTPN5PTPN11MEN1KMT2A
SCHEMBL28510680 0.83 MAPT (0.62) DUSP3PTPN5PTPN11MEN1KMT2A
SCHEMBL28511998 0.83 MAPT (0.61) DUSP3PTPN5PTPN11MEN1KMT2A
SCHEMBL28519354 0.83 KMT2A (0.72) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL12387760 0.81 KMT2A (0.71) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL21211496 0.81 KMT2A (0.71) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL28528684 0.81 SIRT1 (0.80) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL28511869 0.80 MAPT (0.59) DUSP3PTPN5PTPN11MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112079744-B Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2021-07-30 CN disclosed
CN-112079744-A Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2020-12-15 CN disclosed