SCHEMBL28523554

SCHEMBL28523554

N#CCC(=O)Nc1ccc2ncnc(NCCc3ccc(Oc4ccccc4)cc3)c2c1.N#CCC(=O)Nc1ccc2ncnc(NCCc3ccc(Oc4ccccc4)cc3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.58
SRC P12931 1/20 0.58
EGFR P00533 4/20 0.54
AURKA O14965 5/20 0.53
CCNC P24863 2/20 0.52
CDK8 P49336 2/20 0.52
CDKN1A P38936 1/20 0.52
CDK19 Q9BWU1 1/20 0.52
ERBB2 P04626 1/20 0.52
CDK1 P06493 3/20 0.48
HTT P42858 2/20 0.46
GMPS P49915 2/20 0.46
NTRK1 P04629 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28531052 0.83 FYN (0.56) FYNSRCEGFRAURKACCNC
SCHEMBL5499111 0.78 SRC (0.71) FYNSRCEGFRAURKACCNC
SCHEMBL8548720 0.77 HTT (0.69) FYNSRCEGFRCCNCCDK8
SCHEMBL157421 0.77 NFKB1 (0.63) FYNSRCEGFRAURKACCNC
SCHEMBL29350229 0.77 NFKB1 (0.63) FYNSRCEGFRAURKACCNC
SCHEMBL5496069 0.76 SRC (0.68) FYNSRCEGFRAURKACCNC
SCHEMBL8543007 0.76 HTT (0.77) EGFRAURKACCNCCDK8CDKN1A
SCHEMBL28530926 0.74 CCNC (0.57) FYNSRCEGFRCCNCCDK8
SCHEMBL8542891 0.74 HTT (0.54) FYNSRCEGFRAURKACCNC
SCHEMBL12297970 0.73 RNF4 (0.65) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112209875-B 6-amino-4- (4-phenoxyphenethylamino) quinazoline derivative and preparation method and application thereof 绍兴文理学院 2021-11-30 CN disclosed
CN-112209875-A 6-amino-4- (4-phenoxyphenethylamino) quinazoline derivative and preparation method and application thereof 绍兴文理学院 2021-01-12 CN disclosed