SCHEMBL28523650

SCHEMBL28523650

CC1CCN(C(=O)Cc2ccc(C(F)(F)F)cc2)[C@]1(COCc1ccccc1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.43
TACR1 P25103 5/20 0.43
SIGMAR1 Q99720 2/20 0.42
SLC6A5 Q9Y345 1/20 0.39
KMT2A Q03164 2/20 0.39
OPRD1 P41143 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
ME2 P23368 1/20 0.39
ME1 P48163 1/20 0.39
ME3 Q16798 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CCR5 P51681 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
LIPG Q9Y5X9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28523651 1.00 KCNH2 (0.43) KCNH2TACR1SIGMAR1SLC6A5KMT2A
SCHEMBL28907976 0.89 SMN1; SMN2 (0.42) SIGMAR1KMT2AMEN1ALDH1A1
SCHEMBL28907975 0.89 SMN1; SMN2 (0.42) SIGMAR1KMT2AMEN1ALDH1A1
SCHEMBL28991793 0.84 TACR1 (0.42) KCNH2TACR1SIGMAR1SLC6A5LIPG
SCHEMBL28545922 0.77 SMN1; SMN2 (0.38)
SCHEMBL28522821 0.77 TACR1 (0.47) TACR1
SCHEMBL28528445 0.76 CHRM5 (0.42) HRH3
SCHEMBL28528446 0.76 CHRM5 (0.42) HRH3
SCHEMBL28523719 0.74 TACR1 (0.46) TACR1
SCHEMBL28519269 0.74 ALDH1A1 (0.45) KMT2AOPRD1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112174869-A Preparation method and medicinal application of N-phenylacetyl-2-hydroxymethyl pyrrolidine-2-formamide 蔡霈 2021-01-05 CN disclosed