SCHEMBL28525633

SCHEMBL28525633

COC(=O)c1cc(Br)cc(NC2CCCCC2)c1O

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 1/20 0.51
OPRK1 P41145 17/20 0.47
KDM4E B2RXH2 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13276681 0.86 YAP1 (0.54) YAP1OPRK1KDM4E
SCHEMBL13276979 0.85 YAP1 (0.52) YAP1OPRK1KDM4E
SCHEMBL13280433 0.84 OPRK1 (0.48) YAP1OPRK1KDM4E
SCHEMBL4583665 0.82 YAP1 (0.55) YAP1OPRK1KDM4E
SCHEMBL8833932 0.81 YAP1 (0.62) YAP1OPRK1KDM4E
SCHEMBL19391535 0.81 YAP1 (0.48) YAP1OPRK1KDM4EOPRM1OPRD1
SCHEMBL31535175 0.78 YAP1 (0.50) YAP1OPRK1KDM4E
SCHEMBL25194622 0.77 KDM4E (0.56) KDM4E
SCHEMBL15566591 0.74 ABCG2 (0.47) YAP1OPRK1KDM4E
SCHEMBL13277104 0.74 YAP1 (0.41) YAP1OPRK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107573336-B Benzoheterocycle-formamide-pyridone derivative and preparation method and application thereof 四川大学 2021-01-19 CN disclosed