SCHEMBL28525978

SCHEMBL28525978

Cc1cc(N2CCC(c3ccc(C(F)(F)F)cc3)C2)ccc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.51
MAPT P10636 5/20 0.45
ALDH1A1 P00352 3/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
SIRT6 Q8N6T7 1/20 0.44
SERPINE1 P05121 3/20 0.43
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
POLB P06746 1/20 0.42
LMNA P02545 4/20 0.42
TDP1 Q9NUW8 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
NOTUM Q6P988 1/20 0.41
MAPK1 P28482 2/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30474517 1.00 HPGD (0.51) HPGDMAPTALDH1A1MEN1KMT2A
SCHEMBL28532606 0.82 NOTUM (0.49) MAPTALDH1A1MEN1KMT2ASIRT6
SCHEMBL30474439 0.81 NOTUM (0.42) NOTUM
SCHEMBL13884398 0.79 HPGD (0.63) HPGDMAPTALDH1A1KMT2ASIRT6
SCHEMBL14938549 0.79 HPGD (0.63) HPGDMAPTALDH1A1KMT2ASIRT6
SCHEMBL28547071 0.78 ALDH1A1 (0.45) MAPTALDH1A1MEN1KMT2ACYP2C9
SCHEMBL28532287 0.78 CHRNB2 (0.53) MAPTALDH1A1MEN1KMT2ASERPINE1
SCHEMBL21619788 0.77 NOTUM (0.51) MAPTALDH1A1CYP3A4NOTUMRAB9A
SCHEMBL4256964 0.76 HPGD (0.59) HPGDMAPTALDH1A1KMT2ASIRT6
SCHEMBL5388184 0.75 HPGD (0.62) HPGDMAPTALDH1A1KMT2ASIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed