SCHEMBL28532606

SCHEMBL28532606

O=[N+]([O-])c1ccc(N2CCC(c3ccc(C(F)(F)F)cc3)C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.49
ENPP2 Q13822 1/20 0.48
POLB P06746 1/20 0.46
HTR1A P08908 1/20 0.45
MAPT P10636 6/20 0.44
ALDH1A1 P00352 4/20 0.44
LMNA P02545 2/20 0.44
MAPK1 P28482 2/20 0.44
GAA P10253 1/20 0.44
HSD11B1 P28845 2/20 0.44
SLC18A3 Q16572 1/20 0.43
SERPINE1 P05121 1/20 0.43
SLC6A9 P48067 1/20 0.43
SLC6A5 Q9Y345 1/20 0.43
SIRT6 Q8N6T7 2/20 0.43
ADRB1 P08588 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28536975 0.93 MAPT (0.49) NOTUMENPP2POLBHTR1AMAPT
SCHEMBL28532287 0.83 CHRNB2 (0.53) NOTUMPOLBMAPTALDH1A1SERPINE1
SCHEMBL6714666 0.83 MAPT (0.53) POLBHTR1AMAPTALDH1A1LMNA
SCHEMBL30474477 0.82 MAPT (0.55) POLBMAPTALDH1A1LMNAMAPK1
SCHEMBL28537487 0.82 MAPT (0.55) POLBMAPTALDH1A1LMNAMAPK1
SCHEMBL28539978 0.82 ACACB (0.41) POLBMAPTALDH1A1LMNAMAPK1
SCHEMBL30474517 0.82 HPGD (0.51) NOTUMPOLBMAPTALDH1A1LMNA
SCHEMBL28547071 0.82 ALDH1A1 (0.45) MAPTALDH1A1LMNASLC6A9SLC6A5
SCHEMBL28525978 0.82 HPGD (0.51) NOTUMPOLBMAPTALDH1A1LMNA
SCHEMBL21619788 0.80 NOTUM (0.51) NOTUMMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed