SCHEMBL28526410

SCHEMBL28526410

COC(=O)[C@H](Cc1ccccc1)C(C(=O)Cc1ccc(-c2ccccc2)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.47
ITGB7 P26010 2/20 0.47
CTSS P25774 3/20 0.46
CTSK P43235 2/20 0.46
F10 P00742 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
KLK5 Q9Y337 1/20 0.43
HDAC1 Q13547 4/20 0.42
HDAC6 Q9UBN7 4/20 0.42
F2 P00734 2/20 0.42
PRSS1 P07477 2/20 0.42
ACE P12821 2/20 0.42
MME P08473 1/20 0.42
ACE2 Q9BYF1 1/20 0.42
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28540413 0.89 CTSS (0.42) ITGA4ITGB7CTSSCTSKF10
SCHEMBL11382563 0.85 MEN1 (0.53) ITGA4ITGB7CTSSCTSKMEN1
SCHEMBL24404141 0.84 ALDH1A1 (0.44) ITGA4ITGB7CTSSCTSKMEN1
SCHEMBL20583296 0.84 ALDH1A1 (0.44) ITGA4ITGB7CTSSCTSKMEN1
SCHEMBL28538183 0.82 ALDH1A1 (0.42) ITGA4ITGB7CTSSCTSKMEN1
SCHEMBL7415317 0.80 CTSS (0.48) ITGA4ITGB7CTSSCTSKF10
SCHEMBL7415313 0.80 CTSS (0.48) ITGA4ITGB7CTSSCTSKF10
SCHEMBL17871186 0.80 ITGA4 (0.46) ITGA4ITGB7CTSSCTSKMEN1
SCHEMBL20583506 0.78 POLB (0.42) POLB
SCHEMBL24404076 0.78 POLB (0.42) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106977415-B Intermediate of shakubiqu and preparation method thereof 广东东阳光药业有限公司 2021-03-26 CN disclosed