SCHEMBL28526550

SCHEMBL28526550

c1ccc2sc(C3CCCN3)cc2c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
NR1H4 Q96RI1 1/20 0.40
CHRM5 P08912 3/20 0.39
CHRM3 P20309 3/20 0.39
CHRM1 P11229 2/20 0.39
CHRM2 P08172 2/20 0.39
CHRM4 P08173 2/20 0.39
ALOX5 P09917 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7865136 0.95 SLC6A4 (0.43) SLC6A4DRD2HTR2AHTR2CNR1H4
SCHEMBL10571544 0.94 SLC6A4 (0.42) SLC6A4DRD2HTR2AHTR2CNR1H4
SCHEMBL7993434 0.79 HTR2A (0.40) SLC6A4DRD2HTR2AHTR2CCHRM5
Hydrochloric Acid SCHEMBL8688971 0.78 HTR2A (0.42) SLC6A4DRD2HTR2AHTR2CCHRM5
SCHEMBL31172103 0.75 SLC6A4 (0.61) SLC6A4DRD2CHRM5CHRM3CHRM1
SCHEMBL28359596 0.75 SLC6A4 (0.61) SLC6A4DRD2CHRM5CHRM3CHRM1
SCHEMBL2708963 0.75 SLC6A4 (0.54) SLC6A4DRD2HTR2AHTR2CNR1H4
SCHEMBL6685675 0.72 ALOX5 (0.43) SLC6A4DRD2HTR2AHTR2CALOX5
SCHEMBL14559239 0.72 SLC6A4 (0.42) SLC6A4DRD2HTR2AHTR2CCHRM5
SCHEMBL31412580 0.71 SLC6A4 (0.50) SLC6A4DRD2HTR2AHTR2CCHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683029-A Bcl-2 inhibitors 百济神州有限公司 2024-03-12 CN disclosed
CN-117430601-A Bcl-2 inhibitors 百济神州有限公司 2024-01-23 CN disclosed
CN-112437772-B Bcl-2 inhibitors 百济神州有限公司 2023-11-21 CN disclosed
CN-112010859-B Fused ring compound, preparation method and application thereof 中国科学院上海药物研究所 2022-07-19 CN disclosed
CN-112437772-A Bcl-2 inhibitors 百济神州有限公司 2021-03-02 CN disclosed
CN-112010859-A Fused ring compound, preparation method and application thereof 中国科学院上海药物研究所 2020-12-01 CN disclosed