SCHEMBL7865136

SCHEMBL7865136

c1ccc2sc(C3CCCCN3)cc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.43
DRD2 P14416 1/20 0.43
NR1H4 Q96RI1 2/20 0.41
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
MEN1 O00255 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2A6 P11509 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX5 P09917 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10571544 0.98 SLC6A4 (0.42) SLC6A4DRD2NR1H4HTR2AHTR2C
SCHEMBL28526550 0.95 SLC6A4 (0.43) SLC6A4DRD2NR1H4HTR2AHTR2C
SCHEMBL7993434 0.78 HTR2A (0.40) SLC6A4DRD2HTR2AHTR2CCYP2D6
Hydrochloric Acid SCHEMBL8688971 0.77 HTR2A (0.42) SLC6A4DRD2HTR2AHTR2CCYP2D6
SCHEMBL31172103 0.74 SLC6A4 (0.61) SLC6A4DRD2CYP2A6ALOX5SLC6A2
SCHEMBL28359596 0.74 SLC6A4 (0.61) SLC6A4DRD2CYP2A6ALOX5SLC6A2
SCHEMBL2708963 0.73 SLC6A4 (0.54) SLC6A4DRD2NR1H4HTR2AHTR2C
SCHEMBL1257399 0.72 POLB (0.53) CYP2D6CYP2C19POLBCHRNA7CYP1A2
SCHEMBL1257011 0.72 POLB (0.53) CYP2D6CYP2C19POLBCHRNA7CYP1A2
SCHEMBL6685675 0.71 ALOX5 (0.43) SLC6A4DRD2HTR2AHTR2CCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed