SCHEMBL7993434

SCHEMBL7993434

c1ccc2sc(C3CNCCN3)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
SLC6A4 P31645 3/20 0.40
DRD2 P14416 1/20 0.40
SLC6A2 P23975 2/20 0.38
SLC6A3 Q01959 2/20 0.38
ALOX5 P09917 1/20 0.38
CYP2A6 P11509 3/20 0.34
ASIC3 Q9UHC3 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
MGLL Q99685 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
SIGMAR1 Q99720 2/20 0.33
BCL2L1 Q07817 1/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
CYP2D6 P10635 1/20 0.33
PARP1 P09874 1/20 0.33
CHRM2 P08172 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8688971 0.98 HTR2A (0.42) HTR2AHTR2CSLC6A4DRD2SLC6A2
SCHEMBL7993392 0.82 HTR2C (0.36) HTR2AHTR2CSLC6A4SLC6A2SLC6A3
SCHEMBL7997135 0.81 HTR2C (0.37) HTR2AHTR2CSLC6A4SLC6A2ROCK2
SCHEMBL28526550 0.79 SLC6A4 (0.43) HTR2AHTR2CSLC6A4DRD2SLC6A2
SCHEMBL7865136 0.78 SLC6A4 (0.43) HTR2AHTR2CSLC6A4DRD2SLC6A2
SCHEMBL10571544 0.77 SLC6A4 (0.42) HTR2AHTR2CSLC6A4DRD2SLC6A2
SCHEMBL9411183 0.77 CYP2A6 (0.40) CYP2A6ROCK2ROCK1PARP1
Hydrochloric Acid SCHEMBL2957747 0.76 HTR2C (0.36) HTR2AHTR2C
SCHEMBL31412580 0.76 SLC6A4 (0.50) HTR2AHTR2CSLC6A4DRD2SLC6A2
SCHEMBL2708963 0.73 SLC6A4 (0.54) HTR2AHTR2CSLC6A4DRD2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed
US-5136037-A 3-(4-substituted-4-piperazinyl)butyl-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-08-04 US disclosed
US-5037984-A Anticonvulsants; anxiolytic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-06 US disclosed
US-4933453-A ANTIPSYCHOTIC, ANALGESIC, ANTICONVULSANT, AND ANXIOLYTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-12 US disclosed