SCHEMBL28526753

SCHEMBL28526753

CC(C)(C)OC(=O)c1cc(Br)cnc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.38
AAK1 Q2M2I8 1/20 0.37
POLB P06746 1/20 0.36
RORC P51449 1/20 0.36
ALDH1A1 P00352 1/20 0.35
OPRK1 P41145 5/20 0.35
GABRA1 P14867 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35
GABRA4 P48169 2/20 0.35
GABRA6 Q16445 2/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRE P78334 1/20 0.35
GABRG1 Q8N1C3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21596480 0.84 OPRK1 (0.39) ATRAAK1POLBRORCALDH1A1
SCHEMBL18044633 0.83 AAK1 (0.38) AAK1ALDH1A1OPRK1GABRA1GABRG2
SCHEMBL733159 0.82 OPRK1 (0.49) OPRK1
SCHEMBL28528395 0.81 GABRG2 (0.41) ATRPOLBALDH1A1OPRK1GABRA1
SCHEMBL3540698 0.80 AAK1 (0.41) AAK1ALDH1A1OPRK1GABRA1GABRG2
SCHEMBL17315745 0.79 ATR (0.36) ATRPOLBALDH1A1GABRA1GABRG2
SCHEMBL28621778 0.79 ALDH1A1 (0.35) POLBALDH1A1OPRK1
SCHEMBL10324630 0.78 CNR1 (0.38) ATRAAK1POLBALDH1A1GABRA1
SCHEMBL28535766 0.78 OPRK1 (0.48) POLBALDH1A1OPRK1GABRA1GABRG2
SCHEMBL16077093 0.78 OPRK1 (0.40) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112334457-A Process for preparing tricyclic compounds 拜耳公司 2021-02-05 CN disclosed