SCHEMBL2852746

SCHEMBL2852746

CC1CCN(C(c2ccc(F)cc2)c2ccc([C@]3(C(=O)O)CCC3I)cc2-c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.67
PTGS1 P23219 1/20 0.67
PTGS2 P35354 1/20 0.67
PSEN1 P49768 1/20 0.67
PSEN2 P49810 1/20 0.67
APH1B Q8WW43 1/20 0.67
NCSTN Q92542 1/20 0.67
APH1A Q96BI3 1/20 0.67
PSENEN Q9NZ42 1/20 0.67
APP P05067 1/20 0.37
DPP4 P27487 6/20 0.36
DPP7 Q9UHL4 6/20 0.36
DPP8 Q6V1X1 4/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
AKR1C3 P42330 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2849874 0.86 KCNH2 (0.70) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL2849438 0.86 KCNH2 (0.70) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL2846664 0.81 KCNH2 (1.00) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL2847511 0.81 KCNH2 (1.00) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL24913685 0.81 KCNH2 (1.00) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL2846733 0.80 KCNH2 (0.61) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL2850196 0.80 KCNH2 (0.59) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL2844400 0.78 KCNH2 (0.72) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL2850251 0.77 KCNH2 (0.57) KCNH2PTGS1PTGS2PSEN1PSEN2
SCHEMBL2850142 0.77 KCNH2 (0.72) KCNH2PTGS1PTGS2PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010138901-A1 CARBOXYLIC ACID-CONTAINING COMPOUNDS, DERIVATIVES THEREOF, AND RELATED METHODS OF USE BIOGEN IDEC MA INC (US) 2010-12-02 WO claimed