SCHEMBL2852807

SCHEMBL2852807

CC(O)CNS(=O)(=O)c1cccc(C(N)=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.48
PRSS1 P07477 2/20 0.48
PRSS2 P07478 2/20 0.48
PRSS3 P35030 2/20 0.48
F10 P00742 1/20 0.48
CYP2C19 P33261 1/20 0.48
F2 P00734 2/20 0.47
HDAC2 Q92769 2/20 0.47
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
MEP1B Q16820 2/20 0.46
MAPK1 P28482 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032586 0.90 TDP1 (0.50) PRSS1PRSS2PRSS3F10CYP2C19
SCHEMBL28335414 0.83 F2 (0.47) CYP2C19F2HDAC2HDAC8HDAC6
SCHEMBL2850555 0.82 LMNA (0.53) PRSS1PRSS2PRSS3CYP2C19F2
SCHEMBL2852808 0.81 CYP19A1 (0.57) BRAFPRSS1PRSS2PRSS3F2
SCHEMBL3649154 0.80 PTPN11 (0.57) PRSS1PRSS2PRSS3CYP2C19F2
SCHEMBL5041380 0.79 CYP2C19 (0.49) PRSS1PRSS2PRSS3CYP2C19F2
SCHEMBL5034887 0.78 CYP2C19 (0.76) PRSS1PRSS2PRSS3F10CYP2C19
SCHEMBL2859691 0.78 CYP2C19 (0.55) PRSS1PRSS2PRSS3F10CYP2C19
SCHEMBL28208130 0.78 ADAMTS4 (0.50) PRSS1PRSS2PRSS3F10CYP2C19
SCHEMBL2854385 0.77 LMNA (0.56) PRSS1PRSS2PRSS3F2HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed