SCHEMBL28529352

SCHEMBL28529352

O=c1c2cc(Br)ccc2sc2cc3c(=O)c4cc(Br)ccc4sc3cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
EPM2A O95278 1/20 0.45
PTPN2 P17706 1/20 0.45
PTPN1 P18031 1/20 0.45
PTPN22 Q9Y2R2 1/20 0.45
MAPT P10636 4/20 0.42
TP53 P04637 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
RAB9A P51151 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP2A6 P11509 2/20 0.42
HSP90AA1 P07900 1/20 0.40
TLR9 Q9NR96 1/20 0.40
MIF P14174 1/20 0.39
PIM1 P11309 2/20 0.38
CHEK1 O14757 1/20 0.38
AURKA O14965 1/20 0.38
DAPK3 O43293 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5019781 0.96 KDM4E (0.48) KDM4EEPM2APTPN2PTPN1PTPN22
SCHEMBL29466898 0.96 KDM4E (0.48) KDM4EEPM2APTPN2PTPN1PTPN22
SCHEMBL30593470 0.92 KDM4E (0.47) KDM4EEPM2APTPN2PTPN1PTPN22
SCHEMBL18261966 0.92 KDM4E (0.47) KDM4EEPM2APTPN2PTPN1PTPN22
SCHEMBL12811607 0.87 EPM2A (0.50) EPM2APTPN2PTPN1PTPN22MAPT
SCHEMBL1615357 0.86 KDM4E (0.64) KDM4EEPM2APTPN2PTPN1PTPN22
SCHEMBL15226874 0.85 MAPT (0.43) KDM4EEPM2APTPN2PTPN1PTPN22
SCHEMBL18267526 0.85 KDM4E (0.45) KDM4EEPM2APTPN2PTPN1PTPN22
SCHEMBL20383998 0.84 KDM4E (0.42) KDM4EEPM2APTPN2PTPN1PTPN22
SCHEMBL6558940 0.84 KDM4E (0.61) KDM4EEPM2APTPN2PTPN1PTPN22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112390811-B Dithia-anthrone derivative and preparation method and application thereof 中国科学院理化技术研究所 2022-03-04 CN disclosed
CN-112390811-A Dithia-anthrone derivative and preparation method and application thereof 中国科学院理化技术研究所 2021-02-23 CN disclosed