SCHEMBL28529397

SCHEMBL28529397

CC12CCCC(C(=O)Nc3nc4cc(Cl)cc(Cl)c4s3)(CCC1)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.39
CNR1 P21554 1/20 0.38
CCNE1 P24864 5/20 0.38
CDK2 P24941 5/20 0.38
CDK3 Q00526 5/20 0.38
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LCK P06239 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CDK1 P06493 2/20 0.36
CCNB1 P14635 2/20 0.36
GRK2 P25098 2/20 0.35
AURKA O14965 1/20 0.35
FFAR2 O15552 3/20 0.35
DYRK1A Q13627 1/20 0.34
FSCN1 Q16658 1/20 0.34
FPR2 P25090 1/20 0.34
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30944292 1.00 ADORA1 (0.39) ADORA1CNR1CCNE1CDK2CDK3
SCHEMBL30944315 0.85 P2RX7 (0.47) CNR1NPC1RAB9AKMT2ACNR2
SCHEMBL30944357 0.82 ADORA1 (0.56) ADORA1CCNE1CDK2CDK3NPC1
SCHEMBL28523749 0.81 ADORA1 (0.55) ADORA1CCNE1CDK2CDK3NPC1
SCHEMBL30944297 0.81 ADORA1 (0.55) ADORA1CCNE1CDK2CDK3NPC1
SCHEMBL28512789 0.81 DYRK1A (0.58) NPC1RAB9AMEN1KMT2ADYRK1A
SCHEMBL30944286 0.81 DYRK1A (0.58) NPC1RAB9AMEN1KMT2ADYRK1A
SCHEMBL30944281 0.81 NPC1 (0.55) ADORA1CNR1NPC1RAB9AMEN1
SCHEMBL28521684 0.81 NPC1 (0.55) ADORA1CNR1NPC1RAB9AMEN1
SCHEMBL30944284 0.80 NPC1 (0.40) ADORA1CNR1CCNE1CDK2CDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112423746-A Novel anti-mycobacterial heterocyclic amides 克莱斯通公司 2021-02-26 CN claimed
CN-112423746-A Novel anti-mycobacterial heterocyclic amides 克莱斯通公司 2021-02-26 CN disclosed