SCHEMBL28523749

SCHEMBL28523749

CC1(C(=O)Nc2nc3cc(Cl)cc(Cl)c3s2)CCCCCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.55
LCK P06239 1/20 0.45
CYP3A4 P08684 1/20 0.44
PI4KB Q9UBF8 1/20 0.44
CCNE1 P24864 5/20 0.42
CDK2 P24941 5/20 0.42
CDK3 Q00526 5/20 0.42
CDK1 P06493 2/20 0.42
CCNB1 P14635 2/20 0.42
CETP P11597 3/20 0.40
FFAR2 O15552 2/20 0.38
GRK2 P25098 2/20 0.37
AURKA O14965 1/20 0.37
ADORA2A P29274 1/20 0.37
DYRK1A Q13627 1/20 0.37
FSCN1 Q16658 1/20 0.37
NPY2R P49146 1/20 0.36
MEN1 O00255 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30944297 1.00 ADORA1 (0.55) ADORA1LCKCYP3A4PI4KBCCNE1
SCHEMBL30944357 0.99 ADORA1 (0.56) ADORA1LCKCYP3A4PI4KBCCNE1
SCHEMBL30944292 0.81 ADORA1 (0.39) ADORA1LCKCCNE1CDK2CDK3
SCHEMBL28529397 0.81 ADORA1 (0.39) ADORA1LCKCCNE1CDK2CDK3
SCHEMBL30944352 0.80 DYRK1A (0.63) ADORA1LCKDYRK1AFSCN1MEN1
SCHEMBL30944326 0.78 ADORA1 (0.55) ADORA1LCKCYP3A4PI4KBCETP
SCHEMBL30944314 0.76 ADORA1 (0.58) ADORA1LCKCYP3A4PI4KBCCNE1
SCHEMBL30944315 0.75 P2RX7 (0.47) NPC1RAB9AKMT2A
SCHEMBL30944373 0.72 ADORA1 (0.98) ADORA1LCKCYP3A4PI4KBADORA2A
SCHEMBL30944341 0.72 ADORA1 (0.80) ADORA1LCKCYP3A4ADORA2ADYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-112423746-A Novel anti-mycobacterial heterocyclic amides 克莱斯通公司 2021-02-26 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed