SCHEMBL28529563

SCHEMBL28529563

CC(C)(C)COC(=O)NCc1cnn(Cc2ccc(C(F)(F)F)nc2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 8/20 0.39
PPARD Q03181 1/20 0.39
GLS O94925 1/20 0.39
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39
KCNQ4 P56696 1/20 0.39
KCNQ5 Q9NR82 1/20 0.39
NAMPT P43490 1/20 0.38
GAA P10253 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
PTGES O14684 1/20 0.36
RORC P51449 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21491800 0.89 KLKB1 (0.42) KLKB1PPARDGLSKCNQ3KCNQ2
SCHEMBL24400371 0.88 HDAC3 (0.42) KLKB1PPARDGLSKCNQ3KCNQ2
SCHEMBL30744352 0.88 HDAC3 (0.42) KLKB1PPARDGLSKCNQ3KCNQ2
SCHEMBL21491889 0.83 KLKB1 (0.44) KLKB1PPARDGLSNAMPTTRPV1
Trifluoroacetic Acid SCHEMBL30056789 0.78 PPARD (0.42) KLKB1PPARDGLSKCNQ3KCNQ2
Trifluoroacetic Acid SCHEMBL21492407 0.78 PPARD (0.42) KLKB1PPARDGLSKCNQ3KCNQ2
SCHEMBL21491519 0.78 GLS (0.38) KLKB1PPARDGLSCYP3A4CYP2C9
SCHEMBL28532124 0.76 PPARD (0.39) KLKB1PPARDGLSKCNQ3KCNQ2
SCHEMBL30060309 0.74 HDAC3 (0.46) KLKB1NAMPTGAAALDH1A1
SCHEMBL21492632 0.73 PPARD (0.42) PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-B Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2024-03-12 CN disclosed
CN-112218865-A Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2021-01-12 CN disclosed