SCHEMBL30744352

SCHEMBL30744352

CC(C)(C)OC(=O)NCc1cnn(Cc2ccc(C(F)(F)F)nc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
NCOR2 Q9Y618 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
RORC P51449 1/20 0.41
SCD O00767 1/20 0.41
KLKB1 P03952 4/20 0.41
PPARD Q03181 1/20 0.41
GLS O94925 1/20 0.40
NAMPT P43490 4/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
TAS2R8 Q9NYW2 1/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
KCNQ4 P56696 1/20 0.38
KCNQ5 Q9NR82 1/20 0.38
HDAC10 Q969S8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24400371 1.00 HDAC3 (0.42) HDAC3HDAC8NCOR2L3MBTL1RORC
SCHEMBL21491800 0.90 KLKB1 (0.42) RORCKLKB1PPARDGLSNAMPT
SCHEMBL28529563 0.88 KLKB1 (0.39) RORCKLKB1PPARDGLSNAMPT
SCHEMBL30060309 0.86 HDAC3 (0.46) HDAC3HDAC8NCOR2L3MBTL1SCD
SCHEMBL10263975 0.85 L3MBTL1 (0.50) L3MBTL1GLSNAMPTCA1CA2
SCHEMBL21491889 0.85 KLKB1 (0.44) KLKB1PPARDGLSNAMPT
SCHEMBL21503621 0.83 CA1 (0.42) L3MBTL1PPARDGLSNAMPTCA12
SCHEMBL30057190 0.83 CA1 (0.42) L3MBTL1PPARDGLSNAMPTCA12
SCHEMBL30744381 0.82 SCD (0.42) HDAC3HDAC8NCOR2L3MBTL1SCD
SCHEMBL28532083 0.82 SCD (0.42) HDAC3HDAC8NCOR2L3MBTL1SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-B Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2024-03-12 CN disclosed