SCHEMBL28532124

SCHEMBL28532124

NC(=O)OCc1cnn(Cc2ccc(C(F)(F)F)nc2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 1/20 0.39
KCNQ3 O43525 1/20 0.37
KCNQ2 O43526 1/20 0.37
KCNQ4 P56696 1/20 0.37
KCNQ5 Q9NR82 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.36
MGLL Q99685 1/20 0.36
GRM2 Q14416 1/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
KCNH2 Q12809 1/20 0.35
GPR119 Q8TDV5 1/20 0.35
CSF1R P07333 1/20 0.35
LMNA P02545 2/20 0.34
HSD17B10 Q99714 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
PREP P48147 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28524216 0.82 GAA (0.46) KDM4EALDH1A1LMNAHSD17B10MAPT
SCHEMBL8209503 0.81 KLKB1 (0.45) PPARDGRM2KDM4EALDH1A1KCNH2
SCHEMBL28517068 0.81 PPARD (0.39) PPARDKCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL28908750 0.80 GCGR (0.40) PPARDMRGPRX4KCNH2GPR119
SCHEMBL21503682 0.80 LOXL2 (0.40) PPARDKCNH2LMNAGRIN1GRIN2B
Hydrochloric Acid SCHEMBL21491894 0.79 LMNA (0.41) PPARDKCNH2LMNAGRIN1GRIN2B
Hydrochloric Acid SCHEMBL30744436 0.79 LMNA (0.41) PPARDKCNH2LMNAGRIN1GRIN2B
SCHEMBL28524436 0.78 GRM2 (0.31) GRM2LMNAKLKB1
SCHEMBL21492571 0.78 GRIN1 (0.38) PPARDKDM4EALDH1A1KCNH2CSF1R
SCHEMBL21491889 0.78 KLKB1 (0.44) PPARDNAMPTGLSKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-B Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2024-03-12 CN disclosed
CN-112218865-A Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2021-01-12 CN disclosed