SCHEMBL28533103

SCHEMBL28533103

COC(=O)c1cccc(Cn2cc3c(n2)CN(C(=O)O)C3)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD74 P04233 1/20 0.49
MIF P14174 1/20 0.49
ABHD6 Q9BV23 1/20 0.46
SLC7A5 Q01650 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.44
CYP4F2 P78329 2/20 0.43
CYP4A11 Q02928 2/20 0.43
MAPK10 P53779 1/20 0.42
OPRD1 P41143 1/20 0.41
HIF1A Q16665 1/20 0.41
IDO1 P14902 1/20 0.41
KDM4E B2RXH2 1/20 0.41
FOLH1 Q04609 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GSK3B P49841 1/20 0.40
ADCY10 Q96PN6 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22953708 0.88 CD74 (0.52) CD74MIFABHD6SLC7A5LOXL2
SCHEMBL22953220 0.87 CD74 (0.46) CD74MIFABHD6SLC7A5LOXL2
SCHEMBL28521863 0.85 AADAT (0.54) CD74MIFKDM4EMAPTMEN1
SCHEMBL28525980 0.81 PARP1 (0.39) KDM4EL3MBTL1ALDH1A1KMT2AHSD17B10
SCHEMBL28687357 0.81 L3MBTL1 (0.46) KDM4EL3MBTL1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL28511332 0.81 NAMPT (0.45) KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL28507281 0.81 ALDH1A1 (0.47) KDM4EMAPTL3MBTL1MEN1ALDH1A1
SCHEMBL28528135 0.78 AADAT (0.51) MAPTL3MBTL1MEN1ALDH1A1KMT2A
SCHEMBL29774650 0.77 ALDH1A1 (0.43) KDM4EMAPTL3MBTL1MEN1ALDH1A1
SCHEMBL28531542 0.77 ALDH1A1 (0.43) KDM4EMAPTL3MBTL1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300169-B Pyrrolopyrazole derivative, preparation method and medical application thereof 上海美迪西生物医药股份有限公司 2022-03-04 CN disclosed
CN-112300169-A Pyrrolopyrazole derivative, preparation method and medical application thereof 上海美迪西生物医药股份有限公司 2021-02-02 CN disclosed