SCHEMBL28533463

SCHEMBL28533463

O=C(O)c1ccc(N2CC(c3ccc(C(F)(F)F)cc3)C[C@H]2COCC2CC2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 2/20 0.38
LPL P06858 1/20 0.37
LIPG Q9Y5X9 1/20 0.37
F2R P25116 3/20 0.36
LTA4H P09960 1/20 0.36
KDM2B Q8NHM5 1/20 0.36
NOTUM Q6P988 1/20 0.36
P2RY14 Q15391 5/20 0.36
ADRA2A P08913 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
OPRD1 P41143 1/20 0.36
DRD1 P21728 1/20 0.35
DRD5 P21918 1/20 0.35
ADRA1B P35368 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
CCR2 P41597 1/20 0.35
KCNH2 Q12809 1/20 0.35
PTGER4 P35408 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21616595 0.92 SRD5A2 (0.38) SRD5A2LPLLIPGLTA4HKDM2B
SCHEMBL28526814 0.89 SRD5A2 (0.39) SRD5A2LIPGF2RLTA4HP2RY14
SCHEMBL28542508 0.88 SRD5A2 (0.38) SRD5A2F2RLTA4HNOTUMP2RY14
SCHEMBL28532617 0.87 LIPC (0.40) SRD5A2LIPGF2RLTA4HKDM2B
SCHEMBL28910599 0.87 P2RY14 (0.37) SRD5A2F2RLTA4HKDM2BP2RY14
SCHEMBL28910602 0.87 FPR1 (0.41) SRD5A2F2RLTA4HNOTUMP2RY14
SCHEMBL28533648 0.86 P2RY14 (0.43) SRD5A2LIPGF2RP2RY14CCR2
SCHEMBL28532591 0.86 SRD5A2 (0.36) SRD5A2F2RLTA4HP2RY14ADRA2A
SCHEMBL28537090 0.85 PTGIR (0.40) LPLLIPGF2RP2RY14ADRA2A
SCHEMBL23631891 0.85 SRD5A2 (0.39) SRD5A2F2RLTA4HNOTUMP2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed