SCHEMBL28533467

SCHEMBL28533467

O=C1N=C(Nc2ccccc2Cl)C(Nc2ccccc2Cl)=CC1=NNc1nncs1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.36
CYP1A2 P05177 1/20 0.36
MAPT P10636 4/20 0.35
HPGD P15428 4/20 0.35
KDM4E B2RXH2 2/20 0.35
NPC1 O15118 6/20 0.33
RAB9A P51151 6/20 0.33
KDM1A O60341 1/20 0.33
MAPK10 P53779 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 5/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HTT P42858 3/20 0.32
PKM P14618 2/20 0.32
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28511342 0.88 MAPT (0.34) ALDH1A1MAPTHPGDKDM4ERAB9A
SCHEMBL28528237 0.88 TSHR (0.38) ALDH1A1MAPTHPGDKDM4EMEN1
SCHEMBL28518305 0.83 TAAR1 (0.40) ALDH1A1CYP1A2MAPTHPGDKDM4E
SCHEMBL28512480 0.80 KDM1A (0.34) ALDH1A1CYP1A2MAPTHPGDKDM4E
SCHEMBL28519216 0.77 MEN1 (0.37) ALDH1A1CYP1A2MAPTHPGDKDM4E
SCHEMBL28520004 0.76 MAPT (0.46) ALDH1A1MAPTKDM4ENPC1RAB9A
SCHEMBL28515265 0.74 KMT2A (0.41) ALDH1A1CYP1A2MAPTHPGDKDM4E
SCHEMBL4053458 0.71 TSHR (0.41) ALDH1A1MAPTHPGDKDM4ENPC1
SCHEMBL28910372 0.68 ALDH1A1 (0.37) ALDH1A1CYP1A2MAPTRAB9AMAPK10
SCHEMBL30108082 0.68 ALDH1A1 (0.37) ALDH1A1CYP1A2MAPTRAB9AMAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112225733-B Preparation method of 1,3, 4-thiadiazole pyridine-2-ketone derivative and application of derivative as anti-cancer drug 湖南科技大学 2022-12-09 CN disclosed
CN-112225733-A Preparation method of derivative containing 1,3, 4-thiadiazole pyridine-2-ketone and application of derivative as anti-cancer drug 湖南科技大学 2021-01-15 CN disclosed