SCHEMBL30108082

SCHEMBL30108082

O=C1N=CC=C(Nc2cccc(Cl)c2Cl)C1=NNc1nncs1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPK10 P53779 2/20 0.31
DHODH Q02127 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108085 1.00 ALDH1A1 (0.37) ALDH1A1CYP1A2RAB9ASMN1; SMN2MAPK10
SCHEMBL28910372 1.00 ALDH1A1 (0.37) ALDH1A1CYP1A2RAB9ASMN1; SMN2MAPK10
SCHEMBL28524456 0.83 MAPK10 (0.31) ALDH1A1MAPK10
SCHEMBL30108086 0.83 MAPK10 (0.31) ALDH1A1MAPK10
SCHEMBL28515267 0.80 TAAR1 (0.41) ALDH1A1CYP1A2RAB9ASMN1; SMN2MAPT
SCHEMBL28533467 0.68 ALDH1A1 (0.36) ALDH1A1CYP1A2RAB9ASMN1; SMN2MAPK10
SCHEMBL28528237 0.59 TSHR (0.38) ALDH1A1MAPT
SCHEMBL11347865 0.53 CXCL8 (0.55) ALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL1093774 0.52 PTGES2 (0.51) ALDH1A1CYP1A2
SCHEMBL2229840 0.52 MAPT (0.49) ALDH1A1CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112225733-B Preparation method of 1,3, 4-thiadiazole pyridine-2-ketone derivative and application of derivative as anti-cancer drug 湖南科技大学 2022-12-09 CN disclosed