SCHEMBL4053458

SCHEMBL4053458

O=C1C=C(Nc2ccccc2Cl)C(Nc2ccccc2Cl)=NC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HTT P42858 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
APAF1 O14727 2/20 0.40
TDP2 O95551 2/20 0.40
CASP3 P42574 2/20 0.40
SENP8 Q96LD8 2/20 0.40
SENP7 Q9BQF6 2/20 0.40
SENP6 Q9GZR1 2/20 0.40
CDC25B P30305 1/20 0.40
CASP7 P55210 1/20 0.40
CASP9 P55211 1/20 0.40
CASP6 P55212 1/20 0.40
CASP8 Q14790 1/20 0.40
KMT2A Q03164 3/20 0.38
C1R P00736 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4052749 0.91 MAPT (0.41) TSHRADRA2AADRA2BADRA2CALDH1A1
SCHEMBL4053105 0.91 ALDH1A1 (0.42) TSHRADRA2AADRA2BADRA2CALDH1A1
SCHEMBL4058438 0.83 STAT3 (0.42) ADRA2AADRA2BADRA2CALDH1A1HTT
SCHEMBL4059168 0.75 MAPT (0.50) TSHRALDH1A1HTTL3MBTL1APAF1
SCHEMBL28533467 0.71 ALDH1A1 (0.36) ALDH1A1HTTL3MBTL1APAF1TDP2
SCHEMBL30991483 0.70 MAPT (0.62) ALDH1A1HTTL3MBTL1APAF1TDP2
SCHEMBL16296871 0.70 MAPT (0.62) ALDH1A1HTTL3MBTL1APAF1TDP2
SCHEMBL31498989 0.67 TSHR (0.60) TSHRADRA2AADRA2BADRA2CALDH1A1
SCHEMBL1686517 0.67 TSHR (0.60) TSHRADRA2AADRA2BADRA2CALDH1A1
SCHEMBL4051680 0.66 BLM (0.50) ALDH1A1HTTL3MBTL1TDP2CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547713-B2 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2009-06-16 US disclosed
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2006-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives PTGS2, PTGES2, PTGES TSHR 4772/4885ADRA2A 1108/4885ADRA2B 1029/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.