SCHEMBL28533587

SCHEMBL28533587

N#CCC1(Cc2ccccc2)CNCCN1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.35
SIGMAR1 Q99720 2/20 0.34
SLC6A2 P23975 5/20 0.34
SLC6A4 P31645 5/20 0.34
SLC6A3 Q01959 4/20 0.33
CYP2D6 P10635 3/20 0.33
MGLL Q99685 1/20 0.33
KCNH2 Q12809 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19947615 1.00 KMT2A (0.35) KMT2ASIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL22981731 0.86 HTR2C (0.40) KMT2AMEN1CYP2C19JAK2JAK1
Hydrochloric Acid SCHEMBL20168209 0.83 KMT2A (0.40) KMT2ASIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL28785994 0.80 SIGMAR1 (0.42) KMT2ASIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL81980 0.80 ALDH1A1 (0.39) ALDH1A1JAK2JAK1
SCHEMBL1191157 0.75 KMT2A (0.45) KMT2ASIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL1190778 0.75 KMT2A (0.45) KMT2ASIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL28964629 0.75 KMT2A (0.45) KMT2ASIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL27573516 0.73 L3MBTL1 (0.43) KMT2ASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL15202304 0.73 KMT2A (0.39) KMT2ASIGMAR1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112442029-A Tetrahydropyrido [3,4-d ] pyrimidine derivative and application thereof in medicine 四川海思科制药有限公司 2021-03-05 CN disclosed