SCHEMBL28533715

SCHEMBL28533715

COc1ccc2c(cc3n2CCC3=CC(=O)O)c1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.41
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
KDM4E B2RXH2 3/20 0.40
MAPT P10636 3/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 4/20 0.39
POLB P06746 4/20 0.39
HPGD P15428 3/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
THRB P10828 1/20 0.39
TUBB4A P04350 5/20 0.34
TUBB P07437 5/20 0.34
TUBA3C P0DPH7 5/20 0.34
TUBA1B P68363 5/20 0.34
TUBA4A P68366 5/20 0.34
TUBB4B P68371 5/20 0.34
TUBB3 Q13509 5/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2017593 0.86 ALOX5 (0.39) ALOX5KMT2AMEN1KDM4EMAPT
SCHEMBL2014416 0.69 CLK1 (0.32) ALOX5KMT2AMEN1MAPK1GAA
SCHEMBL2017601 0.69 MCL1 (0.40) KMT2AMEN1MAPTRAB9ANPC1
SCHEMBL28537384 0.67 S1PR1 (0.52)
SCHEMBL4036458 0.66 KDM4E (0.39) KMT2AMEN1KDM4EMAPTRAB9A
SCHEMBL4036453 0.66 KDM4E (0.39) KMT2AMEN1KDM4EMAPTRAB9A
SCHEMBL946033 0.66 NTRK1 (0.35) POLBKDM2B
SCHEMBL18052982 0.63 TUBB1 (0.41) KMT2AMEN1MAPTALDH1A1POLB
SCHEMBL2016666 0.62 S1PR1 (0.41) KMT2AMEN1KDM4EALDH1A1POLB
SCHEMBL18054329 0.62 ALDH1A1 (0.43) MAPTALDH1A1POLBHPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105816453-B Substituted tricyclic acid derivatives as S1P1 receptor agonists for the treatment of autoimmune and inflammatory disorders 艾尼纳制药公司 2021-03-05 CN disclosed