SCHEMBL28533787

SCHEMBL28533787

O=C(O)c1cc(F)ccc1NC(=O)C(Cl)(Cl)Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK2 O95069 1/20 0.52
MPO P05164 1/20 0.48
KEAP1 Q14145 1/20 0.46
FABP3 P05413 1/20 0.46
FABP4 P15090 1/20 0.46
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
DHODH Q02127 4/20 0.44
KDM4E B2RXH2 1/20 0.44
HSD17B10 Q99714 1/20 0.44
RBP4 P02753 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
PTPRC P08575 1/20 0.41
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
PTPRA P18433 1/20 0.41
PTPRB P23467 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1893876 0.85 KCNK2 (0.57) KCNK2MPOKEAP1FABP3FABP4
SCHEMBL9200144 0.79 ALDH1A1 (0.49) ALDH1A1MAPTKDM4E
SCHEMBL252578 0.78 KDM4E (0.65) KCNK2MPOKEAP1FABP3FABP4
SCHEMBL7541890 0.78 KEAP1 (0.55) KCNK2MPOKEAP1FABP3FABP4
SCHEMBL7836703 0.78 PTPN1 (0.65) KCNK2MPOKEAP1FABP3FABP4
SCHEMBL9000255 0.77 FABP3 (0.61) KCNK2MPOKEAP1FABP3FABP4
SCHEMBL14854009 0.76 PDK1 (0.42) ALDH1A1GAAKDM4EGRIK1
SCHEMBL19980681 0.75 KEAP1 (0.60) KCNK2MPOKEAP1FABP3FABP4
SCHEMBL16854334 0.74 KDM4E (0.55) KCNK2MPOKEAP1ALDH1A1GAA
SCHEMBL8484239 0.74 KCNK2 (0.49) KCNK2MPOKEAP1FABP3FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112441989-B Preparation method and application of flumazenil intermediate 5-fluoroisatoic anhydride 江苏恩华药业股份有限公司 2022-05-24 CN disclosed
CN-112441989-A Preparation method and application of flumazenil intermediate 5-fluoroisatoic anhydride 江苏恩华药业股份有限公司 2021-03-05 CN disclosed