SCHEMBL28535451

SCHEMBL28535451

CC(C)(C)OC(=O)NN1CC=Cc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 3/20 0.40
DRD2 P14416 6/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
BCHE P06276 1/20 0.37
EPHX2 P34913 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
NPC1 O15118 1/20 0.34
GAA P10253 1/20 0.34
RAB9A P51151 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA7 P43166 1/20 0.34
CA14 Q9ULX7 1/20 0.34
AKT1 P31749 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30040459 0.78 P2RX4 (0.41) P2RX4KMT2AMEN1
SCHEMBL29380399 0.76 BCHE (0.46) P2RX4BCHE
SCHEMBL5560408 0.76 BCHE (0.46) P2RX4BCHE
SCHEMBL27766280 0.75 DRD2 (0.37) DRD2KMT2AMEN1BCHEEPHX2
SCHEMBL30809492 0.73 P2RX4 (0.38) P2RX4
SCHEMBL9420578 0.73 TGM2 (0.37) P2RX4
SCHEMBL29986227 0.72 DRD2 (0.47) DRD2KMT2AMEN1NFKB1NFKB2
SCHEMBL8472507 0.71 P2RX4 (0.37) P2RX4
SCHEMBL1862101 0.69 DRD2 (0.40) DRD2KMT2AMEN1RAB9AL3MBTL1
SCHEMBL3661398 0.69 MAPK1 (0.50) DRD2KMT2AMEN1BCHEEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307772-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-08-27 CN disclosed
CN-106257976-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-02-02 CN disclosed