SCHEMBL28538441

SCHEMBL28538441

c1ccc(Cc2ccc(-c3nccs3)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.71
LOXL2 Q9Y4K0 1/20 0.62
ADRB2 P07550 3/20 0.62
CYP2A6 P11509 1/20 0.49
LTA4H P09960 1/20 0.47
CYP17A1 P05093 2/20 0.46
CYP11B1 P15538 2/20 0.46
CYP11B2 P19099 2/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.46
CALM1 P0DP23 1/20 0.44
FFAR1 O14842 1/20 0.44
HDAC2 Q92769 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21791658 0.92 LOXL2 (0.71) PDPK1LOXL2ADRB2CYP2A6CYP17A1
SCHEMBL5147639 0.84 PDPK1 (0.91) PDPK1LOXL2ADRB2CYP2A6PTGDR2
2-Phenylthiazole SCHEMBL70646 0.84 PDPK1 (1.00) PDPK1LOXL2ADRB2CYP2A6PTGDR2
2-Phenylthiazole SCHEMBL28319382 0.82 PDPK1 (0.95) PDPK1LOXL2ADRB2CYP2A6PTGDR2
2-Phenylthiazole SCHEMBL10519953 0.82 PDPK1 (0.95) PDPK1LOXL2ADRB2CYP2A6PTGDR2
2-Phenylthiazole SCHEMBL4939218 0.82 PDPK1 (0.95) PDPK1LOXL2ADRB2CYP2A6PTGDR2
2-Phenylthiazole SCHEMBL10667585 0.82 PDPK1 (0.95) PDPK1LOXL2ADRB2CYP2A6PTGDR2
2-Phenylthiazole SCHEMBL27882225 0.82 PDPK1 (0.95) PDPK1LOXL2ADRB2CYP2A6PTGDR2
SCHEMBL722198 0.82 PDPK1 (0.77) PDPK1LOXL2ADRB2CYP2A6PTGDR2
SCHEMBL5533749 0.81 LOXL2 (0.62) PDPK1LOXL2ADRB2CYP2A6LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110204507-B Process for producing 2-aryl-4-alkylthiazole compound 浙江大学 2021-03-02 CN disclosed