SCHEMBL5533749

SCHEMBL5533749

c1csc(Cc2ccc(-c3nccs3)cc2)n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.62
ADRB2 P07550 3/20 0.62
PDPK1 O15530 1/20 0.55
LTA4H P09960 1/20 0.48
CYP2A6 P11509 1/20 0.44
CYP17A1 P05093 2/20 0.42
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
ABL1 P00519 1/20 0.39
BCR P11274 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CARM1 Q86X55 2/20 0.38
PRMT1 Q99873 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21791658 0.88 LOXL2 (0.71) LOXL2ADRB2PDPK1CYP2A6CYP17A1
SCHEMBL722198 0.82 PDPK1 (0.77) LOXL2ADRB2PDPK1CYP2A6ABL1
SCHEMBL28538441 0.81 PDPK1 (0.71) LOXL2ADRB2PDPK1LTA4HCYP2A6
SCHEMBL27468396 0.79 NR1H3 (0.51) LOXL2ADRB2LTA4HSLC6A3
SCHEMBL6821892 0.79 LTA4H (0.49) LOXL2ADRB2LTA4HCYP17A1CYP11B1
SCHEMBL27855068 0.79 CYP2C19 (0.50) LOXL2ADRB2LTA4HCYP17A1CYP11B1
SCHEMBL2973461 0.79 LTA4H (0.49) LOXL2ADRB2LTA4H
SCHEMBL6163997 0.79 CYP17A1 (0.50) LOXL2ADRB2PDPK1LTA4HCYP17A1
SCHEMBL378027 0.79 PDPK1 (0.50) PDPK1LTA4HSLC6A3
SCHEMBL534382 0.77 LOXL2 (1.00) LOXL2ADRB2PDPK1LTA4HCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 169 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4359567-A Thermooxidatively stable articulated p-benzobisoxazole and p-benzobisthiazole polymers THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1982-11-16 US claimed
CN-117431020-A Adhesive tape and preparation method and application thereof 太仓金煜电子材料有限公司 2024-01-23 CN disclosed
EP-1384747-B1 PROCESS FOR PRODUCING COMPOSITE FROM SOLUTION OF RIGID POLYMER AND COMPOSITE FILM TOYO BOSEKI (JP) 2013-01-16 EP disclosed
CN-100357344-C Method for producing composite bodies from rigid polymer solutions and composite film TOYO BOSEKI (JP) 2007-12-26 CN disclosed
US-7208109-B2 Changing the solution to nonflowable by absorbing a coagulant, then solvent extraction, for molding a solution of a liquid crystal polymer, polybenzoxazoles or polybenzothiazoles TOYO BOSEKI KABUSHIKI KAISHA (JP) 2007-04-24 US disclosed
US-20060270299-A1 Ballistic-resistant article and process for making the same TOYO BOSEKI KABUSHIKI KAISHA (JP) 2006-11-30 US disclosed
EP-0804639-B1 PROCESS FOR PREPARING POLYBENZAZOLE FILAMENTS AND FIBER TOYO BOSEKI (JP) 2005-10-05 EP disclosed
US-6824871-B2 FIRST COATED WITH A SUBCOAT OF MIXTURE OF WATER-SOLUBLE EPOXY RESIN WITH A VINYLPYRIDINE-STYRENE-BUTADIENE RUBBER LATEX, THEN COATED IN A CONVENTIONAL RESORCINOL-FORMALDEHYDE LATEX TO YIELD A TWICE-COATED YARN THE GOODYEAR TIRE & RUBBER COMPANY 2004-11-30 US disclosed
CN-1500116-A Process for producing composite from solution of rigid polymer and composite film �����֯��ʽ���� 2004-05-26 CN disclosed
US-20040096658-A1 Subcoat for poly (p-phenylene-2,6-benzobisoxazole) fibers GOODYEAR TIRE & RUBBER COMPANY, THE 2004-05-20 US disclosed
EP-0388803-A2 Thermoplastic compositions containing polybenzoxazole; polybenzothiazole and polybenzimidazole moieties and process for making shaped articles therefrom THE DOW CHEMICAL COMPANY (US) 1990-09-26 EP disclosed
US-4959492-A Process to synthesize AB-PBO monomer and phosphate salts thereof THE DOW CHEMICAL COMPANY (US) 1990-09-25 US disclosed
EP-0368006-A2 Copolymers containing polybenzoxazole polybenzothiazole and polybenzimidazole moieties THE DOW CHEMICAL COMPANY (US) 1990-05-16 EP disclosed
WO-1990003995-A1 COPOLYMERS CONTAINING POLYBENZOXAZOLE, POLYBENZOTHIAZOLE AND POLYBENZIMIDAZOLE MOIETIES THE DOW CHEMICAL COMPANY (US) 1990-04-19 WO disclosed
US-4762908-A Polybenzoxazole from aryloxy-2,6-naphthalicdiacid THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1988-08-09 US disclosed
US-4723013-A Aryloxy-2,6-naphthalicdiacid compositions and products produced thereby THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1988-02-02 US disclosed
US-4709006-A Polybenzobisthiazole from aryloxy naphthalic diacid THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1987-11-24 US disclosed
US-4359567-A Thermooxidatively stable articulated p-benzobisoxazole and p-benzobisthiazole polymers THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1982-11-16 US disclosed
US-4359567-A Thermooxidatively stable articulated p-benzobisoxazole and p-benzobisthiazole polymers THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1982-11-16 US disclosed
US-4359567-A Thermooxidatively stable articulated p-benzobisoxazole and p-benzobisthiazole polymers THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1982-11-16 US disclosed