SCHEMBL28538876

SCHEMBL28538876

Cc1nc(OCC2CCCN2C)nc(N2CCN(C(=O)O)CC2)c1Br

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KRAS P01116 9/20 0.44
CHRNB2 P17787 4/20 0.39
CHRNA4 P43681 4/20 0.39
CHRNB4 P30926 2/20 0.39
CHRNA3 P32297 2/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB3 Q05901 1/20 0.39
CHRNA7 P36544 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28538875 1.00 KRAS (0.44) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL22720353 0.88 KRAS (0.44) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL22720351 0.88 KRAS (0.44) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL22720285 0.88 KRAS (0.42) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL28531667 0.86 KRAS (0.45) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL28531666 0.86 KRAS (0.45) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL22720289 0.85 KRAS (0.40) KRAS
SCHEMBL28710948 0.82 KRAS (0.46) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL28710949 0.82 KRAS (0.46) KRASCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL28692003 0.81 KRAS (0.55) KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396147-B Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-06-18 CN disclosed
CN-112552294-B Piperazine heterocyclic derivative-containing inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-19 CN disclosed
CN-113396147-A Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-14 CN disclosed
CN-112552294-A Piperazine heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-03-26 CN disclosed