SCHEMBL28539672

SCHEMBL28539672

CS(=O)(=O)c1ccc(OCC2(CF)CC2)c(C=O)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.38
PTGS1 P23219 1/20 0.38
ERN1 O75460 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
BRD4 O60885 4/20 0.35
GPR119 Q8TDV5 2/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.33
DRD1 P21728 1/20 0.33
ALDH1A1 P00352 2/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
EPAS1 Q99814 1/20 0.32
MAPT P10636 1/20 0.32
PNMT P11086 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28542683 0.95 PTGS2 (0.36) PTGS2PTGS1ERN1SMN1; SMN2BRD4
SCHEMBL28911180 0.88 PTGDR2 (0.38) PTGS2PTGS1ERN1SMN1; SMN2BRD4
SCHEMBL28549312 0.83 BRD4 (0.47) PTGS2PTGS1ERN1SMN1; SMN2BRD4
SCHEMBL28539709 0.83 PTGDR2 (0.37) PTGS2PTGS1ERN1SMN1; SMN2BRD4
SCHEMBL28911175 0.81 SCN9A (0.42) PTGS2PTGS1ERN1SMN1; SMN2BRD4
SCHEMBL28064700 0.75 PTGS2 (0.44) PTGS2PTGS1ERN1SMN1; SMN2PTGDR2
SCHEMBL9825441 0.72 SMN1; SMN2 (0.40) ERN1SMN1; SMN2PTGDR2ALDH1A1HPGD
SCHEMBL7092074 0.72 SMN1; SMN2 (0.61) PTGS2ERN1SMN1; SMN2ALDH1A1HPGD
SCHEMBL8161041 0.71 PTGER1 (0.48) ERN1SMN1; SMN2PTGDR2ALDH1A1HPGD
SCHEMBL28543000 0.70 PTGS2 (0.40) PTGS2PTGS1DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105712952-B 2-substituted oxy-5-methylsulfonyl phenyl piperazine amide analogue and preparation method and application thereof 上海翰森生物医药科技有限公司 2021-03-26 CN claimed
CN-105712952-B 2-substituted oxy-5-methylsulfonyl phenyl piperazine amide analogue and preparation method and application thereof 上海翰森生物医药科技有限公司 2021-03-26 CN disclosed