SCHEMBL28064700

SCHEMBL28064700

CS(=O)(=O)c1ccc(OCC(F)(F)F)c(C=O)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.44
SLC6A9 P48067 2/20 0.40
KCNH2 Q12809 1/20 0.40
PTGDR2 Q9Y5Y4 3/20 0.40
SLC2A1 P11166 2/20 0.40
EPAS1 Q99814 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PTGS1 P23219 2/20 0.39
ERN1 O75460 1/20 0.39
UGCG Q16739 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
TNNI3K Q59H18 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28911175 0.79 SCN9A (0.42) PTGS2PTGDR2EPAS1SMN1; SMN2PTGS1
SCHEMBL28615535 0.77 ALDH1A1 (0.48) PTGDR2SMN1; SMN2ALDH1A1MEN1HPGD
SCHEMBL9825441 0.77 SMN1; SMN2 (0.40) PTGDR2SMN1; SMN2ERN1ALDH1A1MEN1
SCHEMBL28064698 0.77 SLC6A9 (0.52) PTGS2SLC6A9KCNH2PTGDR2SMN1; SMN2
SCHEMBL7092074 0.77 SMN1; SMN2 (0.61) PTGS2SMN1; SMN2ERN1ALDH1A1HPGD
SCHEMBL23144386 0.77 ALDH1A1 (0.53) PTGS2SLC6A9KCNH2PTGDR2SMN1; SMN2
SCHEMBL15036874 0.77 PTGS2 (0.46) PTGS2SLC6A9KCNH2PTGDR2EPAS1
SCHEMBL29811827 0.76 PTGS2 (0.43) PTGS2SLC6A9KCNH2PTGDR2SMN1; SMN2
SCHEMBL29986886 0.76 SLC6A9 (0.51) SLC6A9KCNH2
SCHEMBL23144752 0.76 PTGS2 (0.43) PTGS2SLC6A9KCNH2PTGDR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105712945-B 2-substituted oxy-5-methylsulfonyl aryl piperazine amide analogue and preparation method and application thereof 上海翰森生物医药科技有限公司 2020-12-01 CN disclosed
CN-105712945-A 2-Substituted-oxy-5-methylsulfonyl aryl piperazine acidamide analogue and preparation method and application thereof 上海翰森生物医药科技有限公司 2016-06-29 CN disclosed