SCHEMBL9825441

SCHEMBL9825441

CS(=O)(=O)c1ccc(OCCCCBr)c(C=O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
ERN1 O75460 2/20 0.39
S1PR3 Q99500 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.38
ALDH1A1 P00352 5/20 0.37
HPGD P15428 2/20 0.37
HTT P42858 2/20 0.37
KDM4E B2RXH2 2/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PKM P14618 1/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
FDPS P14324 1/20 0.35
TUBB1 Q9H4B7 1/20 0.35
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7092074 0.80 SMN1; SMN2 (0.61) SMN1; SMN2ERN1ALDH1A1HPGDHTT
SCHEMBL7400011 0.77 MAPT (0.50) SMN1; SMN2ERN1ALDH1A1HPGDMAPT
SCHEMBL28064700 0.77 PTGS2 (0.44) SMN1; SMN2ERN1PTGDR2ALDH1A1HPGD
SCHEMBL19328399 0.76 ALDH1A1 (0.42) SMN1; SMN2PTGDR2ALDH1A1HPGDHTT
SCHEMBL8161041 0.76 PTGER1 (0.48) SMN1; SMN2ERN1PTGDR2ALDH1A1HPGD
SCHEMBL9825309 0.75 GCK (0.39) SMN1; SMN2PTGDR2ALDH1A1HPGDHTT
SCHEMBL28549312 0.75 BRD4 (0.47) SMN1; SMN2ERN1PTGDR2ALDH1A1HPGD
SCHEMBL9119355 0.75 KDM4E (0.52) SMN1; SMN2ERN1PTGDR2ALDH1A1HPGD
SCHEMBL720372 0.73 CA12 (0.50) ALDH1A1MEN1KMT2A
SCHEMBL5627486 0.73 CYP19A1 (0.48) SMN1; SMN2ERN1ALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0167371-B1 DIHYDROPYRIDINE COMPOUNDS, THEIR PRODUCTION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-03-06 EP disclosed
US-4727082-A CARDIOVASCULAR DISORDERS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1988-02-23 US disclosed
EP-0167371-A2 Dihydropyridine compounds, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1986-01-08 EP disclosed