SCHEMBL2854073

SCHEMBL2854073

O=C(Nc1ccncc1)c1ccnn1-c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.59
TYK2 P29597 3/20 0.55
JAK2 O60674 2/20 0.55
GLS O94925 1/20 0.54
RIPK1 Q13546 1/20 0.53
HTT P42858 2/20 0.51
FLT1 P17948 2/20 0.51
KDR P35968 2/20 0.51
TAAR1 Q96RJ0 1/20 0.50
POLB P06746 1/20 0.50
STAT3 P40763 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
BRAF P15056 1/20 0.49
ALDH1A1 P00352 1/20 0.48
KDM4E B2RXH2 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TSHR P16473 1/20 0.47
MAPK13 O15264 1/20 0.46
MAPK12 P53778 1/20 0.46
MAPK11 Q15759 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28768950 0.92 ROCK1 (0.62) ROCK1GLSHTTSMN1; SMN2BRAF
SCHEMBL13485755 0.80 GLS (0.53) ROCK1GLSPOLBBRAFKDM4E
SCHEMBL25110209 0.78 GLS (0.52) ROCK1GLSPOLBBRAFALDH1A1
SCHEMBL10061796 0.76 RIPK1 (0.54) ROCK1GLSRIPK1HTTPOLB
SCHEMBL856957 0.76 POLB (0.52) ROCK1GLSHTTPOLBSMN1; SMN2
SCHEMBL17311598 0.75 ROCK1 (1.00) ROCK1
SCHEMBL2863502 0.75 ROCK1 (0.54) ROCK1SMN1; SMN2ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL11893514 0.74 POLB (0.50) ROCK1GLSHTTPOLBSMN1; SMN2
SCHEMBL23780341 0.74 NAPRT (0.43) ROCK1GLSKDRPOLBSMN1; SMN2
SCHEMBL10242690 0.73 MAPK1 (0.51) ROCK1GLSHTTPOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed