SCHEMBL28544367

SCHEMBL28544367

CC(C)(C)OC(=O)n1c(CBr)cc2cc(Cl)ccc21.Cc1c(C)n(C(=O)OC(C)(C)C)c2ccc(Cl)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
RAB9A P51151 1/20 0.34
NR1H2 P55055 4/20 0.34
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34
GABRA5 P31644 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
GABRA1 P14867 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
CASP1 P29466 1/20 0.33
HSD17B10 Q99714 1/20 0.33
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4387957 0.89 NR1H2 (0.40) ACLYNR1H2PPARGPPARALMNA
SCHEMBL31666014 0.86 GABRG2 (0.41) ACLYAKR1C3AKR1C2RAB9AGABRG2
SCHEMBL21731846 0.86 GABRG2 (0.41) ACLYAKR1C3AKR1C2RAB9AGABRG2
SCHEMBL18990363 0.79 NR1H2 (0.40) ACLYNR1H2PPARGPPARALMNA
SCHEMBL29631993 0.79 NR1H2 (0.41) ACLYNR1H2PPARGPPARALMNA
SCHEMBL19013549 0.79 NR1H2 (0.41) ACLYNR1H2PPARGPPARALMNA
SCHEMBL31095612 0.77 NR1H2 (0.43) NR1H2OXER1
SCHEMBL31370553 0.77 GABRG2 (0.42) ACLYNR1H2GABRG2GABRB3GABRA5
SCHEMBL28542079 0.76 SIRT1 (0.40) RAB9AGABRG2GABRB3GABRA5GABRA1
SCHEMBL5096665 0.75 L3MBTL1 (0.44) RAB9ANR1H2ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112654354-A 1,3,4, 9-tetrahydro-2H-pyrido [3,4-b ] indole derivative compound and application thereof 菲尼克思药业股份有限公司 2021-04-13 CN disclosed