SCHEMBL28545129

SCHEMBL28545129

CCCC[Sn](CCCC)(CCCC)c1nn(C)c2ncccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.41
PDE4B Q07343 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
ELANE P08246 2/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.37
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
KDM5A P29375 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
MPO P05164 1/20 0.34
NAMPT P43490 1/20 0.34
CFTR P13569 1/20 0.34
PRKCB P05771 1/20 0.33
GSK3B P49841 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
IDH1 O75874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28558723 0.86 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL28554390 0.84 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DELANE
SCHEMBL14737720 0.78 PGR (0.39) HTTCNR1CNR2L3MBTL1MPO
SCHEMBL14738488 0.77 GRM4 (0.35) PDE4APDE4BPDE4CPDE4DCNR1
SCHEMBL1278237 0.70 NOS3 (0.38) MAPTL3MBTL1TDP1
SCHEMBL12329416 0.70 KDM4D (0.45) PDE4APDE4BPDE4CPDE4DELANE
SCHEMBL31319295 0.70 NOS3 (0.38) MAPTL3MBTL1TDP1
SCHEMBL1671404 0.69 CYP2D6 (0.32) PDE4APDE4BPDE4CPDE4DL3MBTL1
SCHEMBL15913345 0.69 KDM4E (0.33) CNR2L3MBTL1TDP1
SCHEMBL29382435 0.69 CYP2C9 (0.40) L3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109535158-B Bisaryl maleimide compound and pharmaceutically acceptable salt thereof, and preparation method and application thereof 浙江工业大学 2021-04-23 CN disclosed