SCHEMBL28545151

SCHEMBL28545151

COc1ccc(OC(C)=O)c2c(OC)cccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.54
GAA P10253 2/20 0.54
ALDH1A1 P00352 4/20 0.46
KMT2A Q03164 4/20 0.46
POLB P06746 2/20 0.46
KDM4E B2RXH2 2/20 0.46
LMNA P02545 1/20 0.46
PABPC1 P11940 1/20 0.46
XBP1 P17861 1/20 0.46
NFKB1 P19838 1/20 0.46
HTT P42858 1/20 0.46
SMARCA2 P51531 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
TSHR P16473 3/20 0.46
MEN1 O00255 3/20 0.44
PRMT1 Q99873 1/20 0.44
MAPK1 P28482 1/20 0.44
TNFSF11 O14788 1/20 0.43
ESR1 P03372 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11207630 0.85 ESR1 (0.53) MAPTGAAALDH1A1KMT2AKDM4E
SCHEMBL30067054 0.85 ERN1 (0.50) MAPTGAAALDH1A1KMT2APOLB
SCHEMBL11077979 0.83 MAPT (0.63) MAPTGAAALDH1A1KMT2APOLB
SCHEMBL27836294 0.83 TSHR (0.56) MAPTGAAALDH1A1KMT2AKDM4E
SCHEMBL1193308 0.83 KMT2A (0.52) MAPTGAAALDH1A1KMT2APOLB
SCHEMBL9195639 0.82 HTT (0.54) MAPTGAAALDH1A1KMT2AKDM4E
SCHEMBL9629287 0.81 TNFSF11 (0.46) MAPTGAAALDH1A1KMT2APOLB
SCHEMBL9627528 0.81 HTT (0.48) MAPTGAAALDH1A1KMT2APOLB
SCHEMBL27867912 0.80 L3MBTL1 (0.40) MAPTGAAALDH1A1KMT2AKDM4E
SCHEMBL28794942 0.79 ABCB11 (0.47) MAPTGAAALDH1A1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112645809-B Novel coronavirus 3CL protease inhibitor based on menadione structure 上海交通大学 2022-04-26 CN disclosed
CN-112645809-A Novel coronavirus 3CL protease inhibitor based on menadione structure 上海交通大学 2021-04-13 CN disclosed