SCHEMBL28545366

SCHEMBL28545366

COc1ccc(C2=NN(c3ccccc3)C(c3ccc(SC)cc3)C2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.70
ERBB2 P04626 2/20 0.70
L3MBTL1 Q9Y468 5/20 0.69
ATM Q13315 4/20 0.69
RAB9A P51151 1/20 0.69
MEN1 O00255 5/20 0.68
KMT2A Q03164 5/20 0.68
KDM4E B2RXH2 3/20 0.68
ALDH1A1 P00352 3/20 0.68
MAPT P10636 3/20 0.68
LMNA P02545 1/20 0.68
PDE5A O76074 6/20 0.64
USP2 O75604 1/20 0.64
TDP1 Q9NUW8 1/20 0.64
GLA P06280 2/20 0.62
GAA P10253 2/20 0.62
NPSR1 Q6W5P4 2/20 0.62
POLB P06746 1/20 0.62
CDC42 P60953 1/20 0.62
CA1 P00915 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10362296 0.92 EGFR (0.81) EGFRERBB2L3MBTL1ATMRAB9A
SCHEMBL28573013 0.89 EGFR (0.61) EGFRERBB2L3MBTL1ATMMEN1
SCHEMBL8171663 0.89 MEN1 (0.83) EGFRERBB2L3MBTL1ATMRAB9A
SCHEMBL9514571 0.89 MEN1 (0.78) EGFRERBB2L3MBTL1ATMRAB9A
SCHEMBL28547411 0.88 MMP2 (0.56) EGFRERBB2L3MBTL1ATMRAB9A
SCHEMBL11205361 0.87 EGFR (0.74) EGFRERBB2L3MBTL1ATMRAB9A
SCHEMBL11210797 0.87 EGFR (0.74) EGFRERBB2L3MBTL1ATMRAB9A
SCHEMBL15301347 0.86 MEN1 (0.82) EGFRERBB2L3MBTL1ATMRAB9A
SCHEMBL15301136 0.86 KDM4E (0.88) EGFRERBB2L3MBTL1ATMRAB9A
SCHEMBL10654063 0.86 MEN1 (0.91) EGFRERBB2L3MBTL1ATMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574110-B Preparation and application of acyl-substituted pyrazoline sulfonium salt derivative 同济大学 2022-04-19 CN disclosed
CN-112574110-A Preparation and application of acyl-substituted pyrazoline sulfonium salt derivative 同济大学 2021-03-30 CN disclosed