SCHEMBL28545490

SCHEMBL28545490

C1=CN(c2ccccn2)CC(Nc2ccccc2)=C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 2/20 0.40
NPSR1 Q6W5P4 2/20 0.38
THRB P10828 1/20 0.38
PLD1 Q13393 1/20 0.36
CSNK2A1 P68400 1/20 0.35
LMNA P02545 1/20 0.34
SMG1 Q96Q15 1/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
PTGS2 P35354 1/20 0.34
MAPK1 P28482 2/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28545492 0.75 LMNA (0.40) KDM4EALDH1A1NPSR1PLD1LMNA
SCHEMBL28545852 0.74 PLD1 (0.41) KDM4EALDH1A1PLD1LMNAGRIN2D
SCHEMBL21258588 0.74 PLD1 (0.41) KDM4EALDH1A1NPSR1PLD1LMNA
SCHEMBL28545491 0.74 SMN1; SMN2 (0.42) KDM4EALDH1A1PLD1GRIN2DGRIN3B
SCHEMBL28541771 0.74 ALDH1A1 (0.39) KDM4EALDH1A1NPSR1PLD1USP2
SCHEMBL28545020 0.71 HTT (0.41) KDM4EALDH1A1PLD1LMNAGRIN2D
SCHEMBL30565007 0.65 PLD1 (0.44) KDM4EALDH1A1PLD1LMNAGRIN2D
SCHEMBL2096767 0.65 PLD1 (0.44) KDM4EALDH1A1PLD1LMNAGRIN2D
SCHEMBL1140766 0.65 PLD1 (0.47) KDM4EALDH1A1PLD1GRIN2DGRIN3B
SCHEMBL5145918 0.64 PLD1 (0.43) KDM4EALDH1A1PLD1LMNAGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109678854-B Method for synthesizing pyrido [1,2-a ] indole-6 (1H) -ketone compound by manganese catalysis 陕西师范大学 2021-04-09 CN disclosed