SCHEMBL2854555

SCHEMBL2854555

COC(=O)[C@H](C)N(C(=O)OC(C)(C)C)c1ccc(-c2cccc3ccccc23)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 11/20 0.45
PPARA Q07869 11/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
PPARD Q03181 1/20 0.45
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
BRD4 O60885 2/20 0.38
PAX8 Q06710 1/20 0.38
CREBBP Q92793 1/20 0.37
MEN1 O00255 1/20 0.36
PLA2G1B P04054 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855837 0.84 ITGA4 (0.39) PPARGPPARABRD4PAX8CREBBP
SCHEMBL7446003 0.84 KMT2A (0.41) CYP2C9CYP2C19BRD4PAX8MEN1
SCHEMBL7308442 0.84 KMT2A (0.41) CYP2C9CYP2C19BRD4PAX8MEN1
SCHEMBL6139113 0.82 MEN1 (0.40) BRD4MEN1PLA2G1BHTTKMT2A
SCHEMBL27597531 0.82 MEN1 (0.40) BRD4MEN1PLA2G1BHTTKMT2A
SCHEMBL8380101 0.81 KMT2A (0.45) MEN1PLA2G1BHTTKMT2ANPSR1
SCHEMBL27597529 0.79 MEN1 (0.42) PPARGPPARAPPARDPAX8MEN1
SCHEMBL6139041 0.79 MEN1 (0.42) PPARGPPARAPPARDPAX8MEN1
SCHEMBL2861381 0.79 XBP1 (0.37) PAX8MEN1PLA2G1BHTTKMT2A
SCHEMBL2855207 0.79 ITGA4 (0.37) BRD4PAX8CREBBPMEN1PLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346971-B1 Production method for biarylalanine SUMITOMO CHEMICAL CO (JP) 2010-01-20 EP disclosed
EP-1346971-A1 Production method for biarylalanine SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2003-09-24 EP disclosed