SCHEMBL2854612

SCHEMBL2854612

CC(NC(=O)c1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F)c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.53
MAPT P10636 3/20 0.48
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TRPC3 Q13507 1/20 0.44
CYP3A4 P08684 4/20 0.43
GPR6 P46095 1/20 0.42
KMT2A Q03164 1/20 0.41
MALT1 Q9UDY8 1/20 0.41
HSD11B1 P28845 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853091 0.90 MAPT (0.49) CCR1MAPTKDM4EALDH1A1POLB
SCHEMBL2858033 0.81 KDM4E (0.58) CCR1MAPTKDM4EALDH1A1POLB
SCHEMBL2856075 0.81 NAMPT (0.56) MAPTKDM4EALDH1A1POLBSMN1; SMN2
SCHEMBL2852992 0.80 CCR1 (0.53) CCR1MAPTKDM4EALDH1A1POLB
SCHEMBL2855462 0.79 MAPT (0.54) CCR1MAPTKDM4EALDH1A1POLB
SCHEMBL2856202 0.78 CCR1 (0.55) CCR1MAPTKDM4EALDH1A1POLB
SCHEMBL2852931 0.77 KDM4E (0.57) CCR1MAPTKDM4EALDH1A1POLB
SCHEMBL2854457 0.77 CYP3A4 (0.43) MAPTPOLBSMN1; SMN2CYP3A4KMT2A
SCHEMBL2860428 0.76 KDM4E (0.52) CCR1MAPTKDM4EALDH1A1POLB
SCHEMBL2855128 0.76 TRPC3 (0.56) CCR1MAPTKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed