SCHEMBL28546191

SCHEMBL28546191

CCN1CCN(c2cc(OC(N)=O)c([N+](=O)[O-])c(C(C)(C)C)c2)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.39
LMNA P02545 5/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 10/20 0.35
KDM4E B2RXH2 2/20 0.35
KMT2A Q03164 2/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.34
HTT P42858 1/20 0.34
TP53 P04637 1/20 0.34
BLM P54132 1/20 0.34
GAA P10253 1/20 0.33
RAD52 P43351 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28539777 0.83 MAPT (0.40) ALDH1A1LMNAMAPTKDM4EKMT2A
SCHEMBL28546189 0.79 MAPT (0.47) ALDH1A1LMNAL3MBTL1CYP2D6MAPT
SCHEMBL28537173 0.78 MAPT (0.55) ALDH1A1LMNAL3MBTL1CYP2D6MAPT
SCHEMBL22321541 0.77 MAPT (0.47) ALDH1A1LMNAL3MBTL1CYP2D6MAPT
SCHEMBL28537399 0.75 MAPT (0.33) L3MBTL1MAPTKMT2ASMN1; SMN2HTT
SCHEMBL21596369 0.72 GAA (0.50) ALDH1A1LMNAMAPTKDM4EKMT2A
SCHEMBL28539775 0.72 ALDH1A1 (0.39) ALDH1A1LMNACYP2D6MAPTKDM4E
SCHEMBL1421217 0.72 ALDH1A1 (0.42) ALDH1A1L3MBTL1MAPTKDM4EKMT2A
SCHEMBL21596314 0.71 GAA (0.58) LMNAMAPTKDM4EKMT2ASMN1; SMN2
SCHEMBL28526641 0.70 KDM4E (0.36) ALDH1A1MAPTKDM4EKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112313207-B Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2023-02-14 CN disclosed
CN-113087671-B Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2022-10-21 CN disclosed
CN-113087671-A Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2021-07-09 CN disclosed
CN-112313207-A Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2021-02-02 CN disclosed