SCHEMBL28526641

SCHEMBL28526641

CN1CCN(c2cc(OC(N)=O)c(N)c(C(C)(C)C)c2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 1/20 0.36
ADRA2C P18825 2/20 0.36
HRH4 Q9H3N8 2/20 0.36
MAPT P10636 3/20 0.36
KMT2A Q03164 2/20 0.36
GAA P10253 2/20 0.36
PTK2B Q14289 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
POLB P06746 1/20 0.36
GFER P55789 1/20 0.36
ESR2 Q92731 1/20 0.36
MEN1 O00255 1/20 0.35
P2RY1 P47900 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
RECQL P46063 1/20 0.35
SIRT6 Q8N6T7 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28532037 0.90 ALDH1A1 (0.36) KDM4EALDH1A1HSD17B10MAPTKMT2A
SCHEMBL28539777 0.86 MAPT (0.40) KDM4EALDH1A1MAPTKMT2AGAA
SCHEMBL28537166 0.82 L3MBTL3 (0.36)
SCHEMBL28526640 0.77 KDM4E (0.45) KDM4EALDH1A1HSD17B10ADRA2CHRH4
SCHEMBL28751702 0.76 MAPT (0.55) KDM4EALDH1A1HSD17B10ADRA2CMAPT
SCHEMBL28392012 0.71 CA1 (0.47) ALDH1A1KMT2AGAAMEN1MAPK1
SCHEMBL28546191 0.70 ALDH1A1 (0.39) KDM4EALDH1A1MAPTKMT2AGAA
SCHEMBL28388910 0.70 NR1H4 (0.36) KDM4EALDH1A1GAAMAPK1
SCHEMBL21596369 0.69 GAA (0.50) KDM4EALDH1A1HSD17B10MAPTKMT2A
SCHEMBL28751714 0.68 SIRT6 (0.70) ALDH1A1MAPTMAPK1SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113087671-B Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2022-10-21 CN disclosed
CN-113087671-A Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2021-07-09 CN disclosed
CN-112313207-A Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2021-02-02 CN disclosed