SCHEMBL28548723

SCHEMBL28548723

Nc1c(N)n(C2(c3ccc(Cl)cc3)CC2)c(S)nc1=O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.32
CTSD P07339 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
HSD11B1 P28845 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28551647 0.85
SCHEMBL28543435 0.76 PNP (0.37) HSD11B1
SCHEMBL17814738 0.69 TNF (0.42) KDM4EMEN1MAPTKMT2ASMN1; SMN2
SCHEMBL18950494 0.59 CDC25A (0.37) MEN1MAPTKMT2ASMN1; SMN2
SCHEMBL1047702 0.59 CDC25A (0.37) MEN1MAPTKMT2ASMN1; SMN2
SCHEMBL1048937 0.57 NPC1 (0.38) MEN1MAPTKMT2ASMN1; SMN2
SCHEMBL27173413 0.56 HDAC4 (0.44) BACE1HSD11B1
SCHEMBL10743825 0.55 CYP19A1 (0.57) HSD11B1KDM4E
SCHEMBL1975025 0.54 HSD11B1 (0.56) HSD11B1KDM4EKMT2ASMN1; SMN2
SCHEMBL5253993 0.53 CCR2 (0.49) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409331-B Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-20 CN disclosed
CN-112409331-A Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-02-26 CN disclosed