SCHEMBL17814738

SCHEMBL17814738

Nc1c(N)n(Cc2ccc(Cl)cc2)c(S)nc1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.42
CXCL8 P10145 1/20 0.42
SOS1 Q07889 1/20 0.42
NOD2 Q9HC29 1/20 0.42
NOD1 Q9Y239 1/20 0.42
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TYMS P04818 1/20 0.40
GAA P10253 1/20 0.38
GFER P55789 1/20 0.38
TLR7 Q9NYK1 4/20 0.38
TSHR P16473 1/20 0.38
TLR8 Q9NR97 1/20 0.37
POLB P06746 2/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 3/20 0.36
IDO1 P14902 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814737 0.83 ALDH1A1 (0.41) TNFCXCL8SOS1NOD2NOD1
SCHEMBL28547235 0.81 RAB9A (0.45) TNFCXCL8SOS1NOD2NOD1
SCHEMBL28537635 0.79 TSHR (0.37) TNFCXCL8SOS1NOD2NOD1
SCHEMBL17814735 0.73 PNP (0.57) TLR7TLR8KMT2A
SCHEMBL29172435 0.73 P2RX3 (0.42) NOD1GAALMNA
SCHEMBL28548723 0.69 BACE1 (0.32) KDM4ESMN1; SMN2MAPTMEN1KMT2A
SCHEMBL28538573 0.68 ALDH1A1 (0.39) NOD1ALDH1A1KDM4ESMN1; SMN2HPGD
SCHEMBL30804819 0.68 BRD4 (0.42) ALDH1A1KDM4ESMN1; SMN2HPGDHSD17B10
SCHEMBL11719377 0.68 P2RX3 (0.54) ALDH1A1KDM4ESMN1; SMN2TSHRPOLB
SCHEMBL10795638 0.66 CLPP (0.48) TNFCXCL8SOS1NOD2NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409331-B Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-20 CN disclosed
CN-112409331-A Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-02-26 CN disclosed
WO-2017209267-A1 PURINE DERIVATIVE 塩野義製薬株式会社 2017-12-07 WO disclosed
WO-2016088838-A1 PURINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION THEREOF 塩野義製薬株式会社 2016-06-09 WO disclosed