SCHEMBL28549841

SCHEMBL28549841

O=C(O)c1ccccc1Nc1cccc(Br)c1OCC1CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 4/20 0.52
MAPK8 P45983 1/20 0.50
FABP3 P05413 2/20 0.45
FABP5 Q01469 2/20 0.45
TAS2R14 Q9NYV8 2/20 0.44
SIRT2 Q8IXJ6 1/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
PTGS2 P35354 2/20 0.43
AKR1C3 P42330 2/20 0.43
HIF1A Q16665 2/20 0.43
AKR1B10 O60218 1/20 0.43
TRPA1 O75762 1/20 0.43
ABCB11 O95342 1/20 0.43
DHFR P00374 1/20 0.43
MPO P05164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30462500 1.00 FABP4 (0.52) FABP4MAPK8FABP3FABP5TAS2R14
SCHEMBL30462447 0.85 PBRM1 (0.54) FABP4MAPK8FABP3FABP5SIRT2
SCHEMBL28553681 0.85 PBRM1 (0.54) FABP4MAPK8FABP3FABP5SIRT2
SCHEMBL3398683 0.84 THRA (0.45) FABP4MAPK8CXCR5KDM4EKDM5A
SCHEMBL28557288 0.81 MAPK8 (0.53) FABP4MAPK8FABP3FABP5SIRT2
SCHEMBL30462481 0.81 MAPK8 (0.56) FABP4MAPK8FABP3FABP5SIRT2
SCHEMBL30462462 0.81 MAPK8 (0.53) FABP4MAPK8FABP3FABP5SIRT2
SCHEMBL28563343 0.81 MAPK8 (0.56) FABP4MAPK8FABP3FABP5SIRT2
SCHEMBL28559723 0.81 MAPK8 (0.46) FABP4MAPK8FABP3FABP5TAS2R14
SCHEMBL30462460 0.81 MAPK8 (0.46) FABP4MAPK8FABP3FABP5TAS2R14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112745237-B 2-arylamine compound and preparation method and application thereof 中国科学院上海药物研究所 2023-06-20 CN disclosed
CN-112745237-A 2-arylamine compound and preparation method and application thereof 中国科学院上海药物研究所 2021-05-04 CN disclosed