SCHEMBL28550577

SCHEMBL28550577

CCOC(=O)c1nccc(Br)c1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.47
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 2/20 0.44
HPGD P15428 1/20 0.44
CYP1A2 P05177 3/20 0.44
LMNA P02545 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAOA P21397 1/20 0.44
TARBP2 Q15633 1/20 0.42
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NUDT1 P36639 1/20 0.40
CDC7 O00311 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
ALOX15 P16050 2/20 0.40
TSHR P16473 2/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28634780 0.84 BRD4 (0.49) BRD4ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL30662586 0.84 BRD4 (0.49) BRD4KDM4ECYP1A2TARBP2MAPT
SCHEMBL14895438 0.83 BRD4 (0.48) BRD4ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL25347956 0.83 BRD4 (0.48) BRD4ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL15758316 0.83 NUDT1 (0.51) BRD4ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL5847015 0.81 BRD4 (0.47) BRD4KDM4ECYP1A2TARBP2MAPT
SCHEMBL27510506 0.80 DPP4 (0.47) BRD4ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL7433335 0.79 BRD4 (0.45) BRD4ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL27167369 0.79 BRD4 (0.45) BRD4KDM4ECYP1A2TARBP2MAPT
SCHEMBL23923034 0.78 MAPT (0.47) ALDH1A1KDM4EHSD17B10HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112654621-A Substituted naphthyridinone compounds useful as T cell activators 百时美施贵宝公司 2021-04-13 CN disclosed