SCHEMBL2855247

SCHEMBL2855247

O=C(NCc1ccc(Cl)c(Cl)c1)c1cnn(-c2ccccc2[N+](=O)[O-])c1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.49
MALT1 Q9UDY8 13/20 0.45
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
DDR1 Q08345 1/20 0.42
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
DDR2 Q16832 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42
MAP3K20 Q9NYL2 1/20 0.42
MAP3K2 Q9Y2U5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2848347 0.88 GAA (0.51) CCR1MALT1CYP1A2CYP3A4HPGD
SCHEMBL2859043 0.86 CCR1 (0.62) CCR1MALT1HPGDMAPK14
SCHEMBL2860320 0.86 CCR1 (0.52) CCR1MALT1
SCHEMBL2859287 0.85 TSHR (0.40) CCR1MALT1
SCHEMBL2860444 0.84 CCR1 (0.60) CCR1DDR1MAPK11MAPK14DDR2
SCHEMBL2857636 0.83 KDM4E (0.61) CCR1HPGDDDR1MAPK11MAPK14
SCHEMBL2850536 0.82 CCR1 (0.52) CCR1MALT1HPGDDDR1MAPK11
SCHEMBL2854304 0.81 NPC1 (0.49) CCR1HPGDDDR1MAPK11MAPK14
SCHEMBL2854425 0.79 CCR1 (0.60) CCR1HPGDDDR1MAPK11MAPK14
SCHEMBL2860317 0.78 CCR1 (0.62) CCR1HPGDDDR1MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed