SCHEMBL2848347

SCHEMBL2848347

O=C(NCc1ccccc1)c1cnn(-c2ccccc2[N+](=O)[O-])c1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
HTT P42858 1/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CCR1 P32246 3/20 0.49
HPGD P15428 3/20 0.48
DDR1 Q08345 1/20 0.48
MAPK11 Q15759 1/20 0.48
MAPK14 Q16539 1/20 0.48
DDR2 Q16832 1/20 0.48
TMEM97 Q5BJF2 1/20 0.48
MAP3K20 Q9NYL2 1/20 0.48
MAP3K2 Q9Y2U5 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
MALT1 Q9UDY8 3/20 0.44
CNR2 P34972 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859043 0.91 CCR1 (0.62) ALDH1A1CCR1HPGDMAPK14MALT1
SCHEMBL2860320 0.90 CCR1 (0.52) HTTKDM4EALDH1A1CCR1MALT1
SCHEMBL2854304 0.90 NPC1 (0.49) GAAKDM4EALDH1A1CCR1HPGD
SCHEMBL2855247 0.88 CCR1 (0.49) CCR1HPGDDDR1MAPK11MAPK14
SCHEMBL2855062 0.84 CCR1 (0.65) KDM4EALDH1A1CCR1HPGDDDR1
SCHEMBL2856256 0.84 MAPT (0.61) HTTKDM4EALDH1A1MEN1KMT2A
SCHEMBL2863137 0.83 GAA (0.44) GAAHTTCCR1HPGDCYP1A2
SCHEMBL2855124 0.83 KDM4E (0.47) KDM4EALDH1A1KMT2AMALT1MAPT
SCHEMBL2852100 0.82 MAPK11 (0.49) KDM4EALDH1A1DDR1MAPK11MAPK14
SCHEMBL2860213 0.81 KDM4E (0.73) KDM4EALDH1A1CCR1HPGDDDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed